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Synthesis of ([1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)phosphonates and their benzo derivatives via 5-exo-dig cyclization

A series of novel 3-methylphosphonylated [1,2,4]triazolo[4,3-a]pyridines was accessed through a 5-exo-dig-type cyclization of chloroethynylphosphonates and commercially available N-unsubstituted 2-hydrazinylpyridines. In addition, 3-methylphosphonylated [1,2,4]triazolo[4,3-a]quinolines and 1-methylp...

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Dettagli Bibliografici
Pubblicato in:Beilstein J Org Chem
Autori principali: Krylov, Aleksandr S, Petrosian, Artem A, Piterskaya, Julia L, Svintsitskaya, Nataly I, Dogadina, Albina V
Natura: Artigo
Lingua:Inglês
Pubblicazione: Beilstein-Institut 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6633597/
https://ncbi.nlm.nih.gov/pubmed/31354875
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.15.159
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