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High-Throughput Dissolution/Permeation Screening—A 96-Well Two-Compartment Microplate Approach

Early formulation screening can alleviate development of advanced oral drug formulations, such as amorphous solid dispersions (ASDs). Traditionally, dissolution is used to predict ASD performance. Here, a high-throughput approach is described that simultaneously screens drug dissolution and permeati...

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Vydáno v:Pharmaceutics
Hlavní autoři: Jacobsen, Ann-Christin, Krupa, Anna, Brandl, Martin, Bauer-Brandl, Annette
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6572106/
https://ncbi.nlm.nih.gov/pubmed/31083433
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics11050227
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