A carregar...

Importance of the Proximity and Orientation of Ligand-Linkage to the Design of Cinnamate-GW9662 Hybrid Compounds as Covalent PPARγ Agonists

Covalent agonists of PPARγ cause unique receptor conformational changes and behave as selective PPARγ modulators, whereas there are few covalent agonists other than endogenous unsaturated fatty acids metabolites. Previously, we established a cell-based strategy to identify new PPARγ ligands and synt...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Utsugi, Yuki, Kobuchi, Hirona, Kawamura, Yukio, Atito, Ahmed Salahelden Aboelhamd, Nagao, Masaya, Isoda, Hiroko, Miyamae, Yusaku
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6571965/
https://ncbi.nlm.nih.gov/pubmed/31137814
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24102019
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!