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Cu-Mediated Aminoquinoline-Directed Radiofluorination of Aromatic C–H Bonds with K(18)F

This communication describes a Cu-mediated ortho-C–H radiofluorination of aromatic carboxylic acids that are protected as 8-aminoquinoline benzamides. The method uses K(18)F and is compatible with a wide range of functional groups. The reaction is showcased in the high specific activity automated sy...

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Bibliographic Details
Published in:Angew Chem Int Ed Engl
Main Authors: Lee, So Jeong, Makaravage, Katarina J., Brooks, Allen F., Scott, Peter J. H., Sanford, Melanie S.
Format: Artigo
Language:Inglês
Published: 2019
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6476334/
https://ncbi.nlm.nih.gov/pubmed/30605563
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201812701
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