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Baricitinib: A 2018 Novel FDA-Approved Small Molecule Inhibiting Janus Kinases

In 2018, Baricitinib was approved by the Food and Drig Administration (FDA) for the treatment of rheumatoid arthritis. Baricitinib exerts its action by targeting Janus kinases (JAK). In this study, we describe the necessary steps for preparing the drug using two alternative routes.

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Bibliographic Details
Published in:Pharmaceuticals (Basel)
Main Authors: Mayence, Annie, Vanden Eynde, Jean Jacques
Format: Artigo
Language:Inglês
Published: MDPI 2019
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6469186/
https://ncbi.nlm.nih.gov/pubmed/30871014
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph12010037
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