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Rational Design, Synthesis and Preliminary Evaluation of Novel Fusarinine C-Based Chelators for Radiolabeling with Zirconium-89

Fusarinine C (FSC) has recently been shown to be a promising and novel chelator for (89)Zr. Here, FSC has been further derivatized to optimize the complexation properties of FSC-based chelators for (89)Zr-labeling by introducing additional carboxylic groups. These were expected to improve the stabil...

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Detalles Bibliográficos
Publicado en:Biomolecules
Autores principales: Zhai, Chuangyan, He, Shanzhen, Ye, Yunjie, Rangger, Christine, Kaeopookum, Piriya, Summer, Dominik, Haas, Hubertus, Kremser, Leopold, Lindner, Herbert, Foster, Julie, Sosabowski, Jane, Decristoforo, Clemens
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6468543/
https://ncbi.nlm.nih.gov/pubmed/30845658
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom9030091
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