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Discovery of 1,4-Naphthoquinones as a New Class of Antiproliferative Agents Targeting GPR55

[Image: see text] A new series of 1,4-naphthoquinones, bearing various cyclic and aliphatic amines on C2, was designed and synthesized to identify antiproliferative agents for triple-negative breast cancer, which represents a clinical challenge without targeted therapies. Among naphthoquinones, 2a a...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Badolato, Mariateresa, Carullo, Gabriele, Caroleo, Maria Cristina, Cione, Erika, Aiello, Francesca, Manetti, Fabrizio
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2019
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6466525/
https://ncbi.nlm.nih.gov/pubmed/30996770
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00333
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