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Resorcinol-, catechol- and saligenin-based bronchodilating β2-agonists as inhibitors of human cholinesterase activity

We investigated the influence of bronchodilating β2-agonists on the activity of human acetylcholinesterase (AChE) and usual, atypical and fluoride-resistant butyrylcholinesterase (BChE). We determined the inhibition potency of racemate and enantiomers of fenoterol as a resorcinol derivative, isoetha...

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Dades bibliogràfiques
Publicat a:J Enzyme Inhib Med Chem
Autors principals: Bosak, Anita, Knežević, Anamarija, Gazić Smilović, Ivana, Šinko, Goran, Kovarik, Zrinka
Format: Artigo
Idioma:Inglês
Publicat: Taylor & Francis 2017
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6445159/
https://ncbi.nlm.nih.gov/pubmed/28573890
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2017.1326109
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