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Simple Entropy Terms for End-Point Binding Free Energy Calculations

We introduce a number of computationally inexpensive modifications to the MM/PBSA and MM/GBSA estimators for binding free energies, which are based on average receptor-ligand interaction energies in simulations of a noncovalent complex, to improve the treatment of entropy: second- and higher-order t...

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Pubblicato in:J Chem Theory Comput
Autori principali: Menzer, William M., Li, Chen, Sun, Wenji, Xie, Bing, Minh, David D. L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6440217/
https://ncbi.nlm.nih.gov/pubmed/30296084
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.8b00418
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