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Probing the Inhibition of Microtubule Affinity Regulating Kinase 4 by N-Substituted Acridones

Microtubule affinity regulating kinase 4 (MARK4) becomes a unique anti-cancer drug target as its overexpression is responsible for different types of cancers. In quest of novel, effective MARK4 inhibitors, some acridone derivatives were synthesized, characterized and evaluated for inhibitory activit...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Voura, Maria, Khan, Parvez, Thysiadis, Savvas, Katsamakas, Sotiris, Queen, Aarfa, Hasan, Gulam Mustafa, Ali, Sher, Sarli, Vasiliki, Hassan, Md. Imtaiyaz
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group UK 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6368574/
https://ncbi.nlm.nih.gov/pubmed/30737440
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-38217-8
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