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Probing the Inhibition of Microtubule Affinity Regulating Kinase 4 by N-Substituted Acridones

Microtubule affinity regulating kinase 4 (MARK4) becomes a unique anti-cancer drug target as its overexpression is responsible for different types of cancers. In quest of novel, effective MARK4 inhibitors, some acridone derivatives were synthesized, characterized and evaluated for inhibitory activit...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Voura, Maria, Khan, Parvez, Thysiadis, Savvas, Katsamakas, Sotiris, Queen, Aarfa, Hasan, Gulam Mustafa, Ali, Sher, Sarli, Vasiliki, Hassan, Md. Imtaiyaz
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6368574/
https://ncbi.nlm.nih.gov/pubmed/30737440
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-38217-8
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