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Efficiency of Stratification for Ensemble Docking using Reduced Ensembles

Molecular docking can account for receptor flexibility by combining the docking score over multiple rigid receptor conformations, such as snapshots from a molecular dynamics simulation. Here, we evaluate a number of common snapshot selection strategies using a quality metric from stratified sampling...

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Bibliografske podrobnosti
izdano v:J Chem Inf Model
Main Authors: Xie, Bing, Clark, John D., Minh, David D. L.
Format: Artigo
Jezik:Inglês
Izdano: 2018
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6338335/
https://ncbi.nlm.nih.gov/pubmed/30114370
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.8b00314
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