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Virtual Screening and Molecular Dynamics Study of Potential Negative Allosteric Modulators of mGluR1 from Chinese Herbs

The metabotropic glutamate subtype 1 (mGluR1), a member of the metabotropic glutamate receptors, is a therapeutic target for neurological disorders. However, due to the lower subtype selectivity of mGluR1 orthosteric compounds, a new targeted strategy, known as allosteric modulators research, is nee...

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Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Jiang, Ludi, Zhang, Xianbao, Chen, Xi, He, Yusu, Qiao, Liansheng, Zhang, Yanling, Li, Gongyu, Xiang, Yuhong
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6332408/
https://ncbi.nlm.nih.gov/pubmed/26184151
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules200712769
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