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Role of BRCA Mutations in Cancer Treatment with Poly(ADP-ribose) Polymerase (PARP) Inhibitors

Inhibition of poly(ADP-ribose) polymerase (PARP) activity induces synthetic lethality in mutated BRCA1/2 cancers by selectively targeting tumor cells that fail to repair DNA double strand breaks (DSBs). Clinical studies have confirmed the validity of the synthetic lethality approach and four differe...

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Dettagli Bibliografici
Pubblicato in:Cancers (Basel)
Autori principali: Faraoni, Isabella, Graziani, Grazia
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6316750/
https://ncbi.nlm.nih.gov/pubmed/30518089
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cancers10120487
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