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Design and Evaluation of a CXCR4 Targeting Peptide 4DV3 as an HIV Entry Inhibitor and a Ligand for Targeted Drug Delivery

The feasibility of utilizing the cell surface chemokine receptor CXCR4 for human immunodeficiency virus (HIV) entry inhibition and as an intracellular portal for targeted drug delivery was evaluated. Novel DV3 ligands (1DV3, 2DV3, and 4DV3) were designed, synthesized and conjugated to various probes...

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Dades bibliogràfiques
Publicat a:Eur J Pharm Biopharm
Autors principals: Lee, In Heon, Palombo, Matthew S., Zhang, Xiaoping, Szekely, Zoltan, Sinko, Patrick J.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6286870/
https://ncbi.nlm.nih.gov/pubmed/29894816
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejpb.2018.06.004
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