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Bioorthogonal Uncaging of the Active Metabolite of Irinotecan by Palladium‐Functionalized Microdevices

SN‐38, the active metabolite of irinotecan, is released upon liver hydrolysis to mediate potent antitumor activity. Systemic exposure to SN‐38, however, also leads to serious side effects. To reduce systemic toxicity by controlling where and when SN‐38 is generated, a new prodrug was specifically de...

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Publicado en:Chemistry
Main Authors: Adam, Catherine, Pérez‐López, Ana M., Hamilton, Lloyd, Rubio‐Ruiz, Belén, Bray, Thomas L., Sieger, Dirk, Brennan, Paul M., Unciti‐Broceta, Asier
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2018
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6282958/
https://ncbi.nlm.nih.gov/pubmed/30187973
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.201803725
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