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Synthesis and SAR Studies of Praziquantel Derivatives with Activity against Schistosoma japonicum

The synthesis and structure-activity relationship (SAR) studies of praziquantel derivatives with activity against adult Schistosoma japonicum are described. Several of them showed better worm killing activity than praziquantel and could serve as leads for further optimization.

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Опубликовано в: :Molecules
Главные авторы: Wang, Wen-Long, Song, Li-Jun, Chen, Xia, Yin, Xu-Ren, Fan, Wen-Hua, Wang, Gu-Ping, Yu, Chuan-Xin, Feng, Bainian
Формат: Artigo
Язык:Inglês
Опубликовано: MDPI 2013
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6269691/
https://ncbi.nlm.nih.gov/pubmed/23912271
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules18089163
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