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Improved Potency and Reduced Toxicity of the Antifungal Peptoid AEC5 Through Submonomer Modification

As proteolytically stable peptidomimetics, peptoids could serve as antifungal agents to supplement a therapeutic field wrought with toxicity issues. We report the improvement of an antifungal peptoid, AEC5, through an iterative structure-activity relationship study. A sarcosine scan was used to firs...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Autores principales: Middleton, Madyson P., Armstrong, Scott A., Bicker, Kevin L.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6246776/
https://ncbi.nlm.nih.gov/pubmed/30297282
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.10.001
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