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New Di-(β-chloroethyl)-α-amides on N-(meta-Acylamino-benzoyl)-D,L-aminoacid Supports with Antitumoral Activity

In order to obtain new compounds with antitumoural action the N-(meta-acylaminobenzoyl)-α-acylaminobenzoyl)-α-aminoacids 4-9 were prepared. These compounds were subsequently converted into the corresponding Δ(2)-oxazolin-5-ones 10-15, which in turn were submitted to a ring opening reaction with di-(...

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Dades bibliogràfiques
Publicat a:Molecules
Autors principals: Sunel, Valeriu, Popa, Marcel, Desbrières, Jacques, Profire, Lenuta, Otilia, Pintilie, Catalina, Lionte
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2008
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6245399/
https://ncbi.nlm.nih.gov/pubmed/18259140
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules13010177
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