Loading...

Kinetic Characterization of Novel HIV-1 Entry Inhibitors: Discovery of a Relationship between Off-Rate and Potency

The entry of HIV-1 into permissible cells remains an extremely attractive and underexploited therapeutic intervention point. We have previously demonstrated the ability to extend the chemotypes available for optimization in the entry inhibitor class using computational means. Here, we continue this...

Full description

Saved in:
Bibliographic Details
Published in:Molecules
Main Authors: Meuser, Megan E., Murphy, Michael B., Rashad, Adel A., Cocklin, Simon
Format: Artigo
Language:Inglês
Published: MDPI 2018
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6222832/
https://ncbi.nlm.nih.gov/pubmed/30081466
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules23081940
Tags: Add Tag
No Tags, Be the first to tag this record!