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Scaffold-Hopping from Synthetic Drugs by Holistic Molecular Representation

The discovery of novel ligand chemotypes allows to explore uncharted regions in chemical space, thereby potentially improving synthetic accessibility, potency, and the drug-likeness of molecules. Here, we demonstrate the scaffold-hopping ability of the new Weighted Holistic Atom Localization and Ent...

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Detalles Bibliográficos
Publicado en:Sci Rep
Main Authors: Grisoni, Francesca, Merk, Daniel, Byrne, Ryan, Schneider, Gisbert
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group UK 2018
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6220272/
https://ncbi.nlm.nih.gov/pubmed/30405170
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-34677-0
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