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Conjugation inhibitors compete with palmitic acid for binding to the conjugative traffic ATPase TrwD, providing a mechanism to inhibit bacterial conjugation

Bacterial conjugation is a key mechanism by which bacteria acquire antibiotic resistance. Therefore, conjugation inhibitors (COINs) are promising compounds in the fight against the spread of antibiotic resistance genes among bacteria. Unsaturated fatty acids (uFAs) and alkynoic fatty acid derivative...

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Dades bibliogràfiques
Publicat a:J Biol Chem
Autors principals: García-Cazorla, Yolanda, Getino, María, Sanabria-Ríos, David J., Carballeira, Néstor M., de la Cruz, Fernando, Arechaga, Ignacio, Cabezón, Elena
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6204903/
https://ncbi.nlm.nih.gov/pubmed/30201608
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA118.004716
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