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Retinal Cholesterol Content Is Reduced in Simvastatin-Treated Mice Due to Inhibited Local Biosynthesis Albeit Increased Uptake of Serum Cholesterol

Statins, a class of cholesterol-lowering drugs, are currently being investigated for treatment of age-related macular degeneration, a retinal disease. Herein, retinal and serum concentrations of four statins (atorvastatin, simvastatin, pravastatin, and rosuvastatin) were evaluated after mice were gi...

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Dettagli Bibliografici
Pubblicato in:Drug Metab Dispos
Autori principali: Mast, Natalia, Bederman, Ilya R., Pikuleva, Irina A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6193214/
https://ncbi.nlm.nih.gov/pubmed/30115644
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.118.083345
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