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Higher ambient synaptic glutamate at inhibitory versus excitatory neurons differentially impacts NMDA receptor activity

Selective disruption of synaptic drive to inhibitory neurons could contribute to the pathophysiology of various brain disorders. We have previously identified a GluN2A-selective positive allosteric modulator, GNE-8324, that selectively enhances N-methyl-d-aspartate receptor (NMDAR)-mediated synaptic...

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Dades bibliogràfiques
Publicat a:Nat Commun
Autors principals: Yao, Lulu, Grand, Teddy, Hanson, Jesse E., Paoletti, Pierre, Zhou, Qiang
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6167324/
https://ncbi.nlm.nih.gov/pubmed/30275542
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-018-06512-7
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