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One Pot Synthesis of α-Aminophosphonates Containing Bromo and 3,4,5-Trimethoxybenzyl Groups under Solvent-free Conditions

New α-aminophosphonates were synthesized by the Kabachnik-Fields reaction of 3,4,5-trimethoxybenzaldehyde (TMB) with p- or m-bromoaniline and a dialkyl phosphite under solvent-free conditions. TMB was prepared from gallic acid via a four step synthetic sequence involving etherification, esterificati...

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Опубликовано в: :Molecules
Главные авторы: Li, Caihong, Song, Baoan, Yan, Kai, Xu, Gangfang, Hu, Deyu, Yang, Song, Jin, Linhong, Xue, Wei, Lu, Ping
Формат: Artigo
Язык:Inglês
Опубликовано: MDPI 2007
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6149498/
https://ncbi.nlm.nih.gov/pubmed/17846566
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/12020163
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