Chargement en cours...

Caffeine inhibition of GLUT1 is dependent on the activation state of the transporter

Caffeine has been shown to be a robust uncompetitive inhibitor of glucose uptake in erythrocytes. It preferentially binds to the nucleotide-binding site on GLUT1 in its tetrameric form and mimics the inhibitory action of ATP. Here we demonstrate that caffeine is also a dose-dependent, uncompetitive...

Description complète

Enregistré dans:
Détails bibliographiques
Publié dans:Biochimie
Auteurs principaux: Gunnink, Leesha K., Busscher, Brianna M., Wodarek, Jeremy A., Rosette, Kylee A., Strohbehn, Lauren E., Looyenga, Brendan D., Louters, Larry L.
Format: Artigo
Langue:Inglês
Publié: 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6141003/
https://ncbi.nlm.nih.gov/pubmed/28322926
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.biochi.2017.03.011
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!