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Vinylation of Benzylic Amines via C–N Bond Functionalization of Benzylic Pyridinium Salts

Cross-couplings of benzylic pyridinium salts and vinylboronic acids or esters have been developed. Via these benzylic pyridinium intermediates, benzylic amines can be engaged in these cross-couplings via C–N bond functionalization. This method boasts mild reaction conditions and excellent tolerance...

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Publicado en:Synthesis (Stuttg)
Autores principales: Guan, Weiye, Liao, Jennie, Watson, Mary P.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6112771/
https://ncbi.nlm.nih.gov/pubmed/30174353
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1055/s-0037-1610084
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