A carregar...

Dissection, Optimization and Structural Analysis of a Covalent Irreversible DDAH1 Inhibitor

Inhibitors of the human enzyme dimethylarginine dimethylaminohydrolase-1 (DDAH1) can control endogenous nitric oxide production. A time-dependent covalent inactivator of DDAH1, N(5)-(1-imino-2-chloroethyl)-l-ornithine (K(I) = 1.3 μM, k(inact) = 0.34 min(−1)), was conceptually dissected into two frag...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Biochemistry
Main Authors: Burstein-Teitelbaum, Gayle, Er, Joyce A.V., Monzingo, Arthur F., Tuley, Alfred, Fast, Walter
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6074031/
https://ncbi.nlm.nih.gov/pubmed/29983043
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b00554
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!