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Towards the rational design of novel drugs based on solubility, partitioning/distribution, biomimetic permeability and biological activity exemplified by 1,2,4-thiadiazole derivatives

Novel 1,2,4-thiadiazole derivatives as potent neuroprotectors were synthesized and identified. Their ability to inhibit the glutamate stimulated Ca(2+) uptake was investigated. The solubility of thiadiazoles was measured in a buffer solution (pH 7.4) at 298 K. The distribution coefficients in 1-octa...

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Detalhes bibliográficos
Publicado no:Medchemcomm
Main Authors: Volkova, T. V., Terekhova, I. V., Silyukov, O. I., Proshin, A. N., Bauer-Brandl, A., Perlovich, G. L.
Formato: Artigo
Idioma:Inglês
Publicado em: Royal Society of Chemistry 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6072304/
https://ncbi.nlm.nih.gov/pubmed/30108702
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6md00545d
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