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Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides

Six tripeptides incorporating acidic amino acid residues were prepared for investigation as activators of β- and γ-carbonic anhydrases (CAs, EC 4.2.1.1) from the pathogenic bacteria Vibrio cholerae, Mycobacterium tuberculosis, and Burkholderia pseudomallei. The primary amino acid residues that are i...

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Bibliografische gegevens
Gepubliceerd in:J Enzyme Inhib Med Chem
Hoofdauteurs: Stefanucci, Azzurra, Angeli, Andrea, Dimmito, Marilisa Pia, Luisi, Grazia, Del Prete, Sonia, Capasso, Clemente, Donald, William A., Mollica, Adriano, Supuran, Claudiu T.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: Taylor & Francis 2018
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6009936/
https://ncbi.nlm.nih.gov/pubmed/29747543
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2018.1468530
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