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Conformational dynamics of P-glycoprotein in lipid nanodiscs and detergent micelles reveal complex motions on a wide time scale

P-glycoprotein (P-gp) is a highly substrate-promiscuous efflux transporter that plays a critical role in drug disposition. P-gp utilizes ATP hydrolysis by nucleotide-binding domains (NBDs) to drive transitions between inward-facing (IF) conformations that bind drugs and outward-facing (OF) conformat...

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Dades bibliogràfiques
Publicat a:J Biol Chem
Autors principals: Li, Mavis Jiarong, Guttman, Miklos, Atkins, William M.
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5925813/
https://ncbi.nlm.nih.gov/pubmed/29511086
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA118.002190
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