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Pharmacokinetic and chemical synthesis optimization of a potent D-peptide HIV entry inhibitor suitable for extended-release delivery

Peptides often suffer from short in vivo half-lives due to proteolysis and renal clearance that limit their therapeutic potential in many indications, necessitating pharmacokinetic (PK) enhancement. D-peptides, composed of mirror-image D-amino acids, overcome proteolytic degradation but are still vu...

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Библиографические подробности
Опубликовано в: :Mol Pharm
Главные авторы: Redman, Joseph S., Francis, J. Nicholas, Marquardt, Robert, Papac, Damon, Mueller, Alan L., Eckert, Debra M., Welch, Brett D., Kay, Michael S.
Формат: Artigo
Язык:Inglês
Опубликовано: 2018
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5893306/
https://ncbi.nlm.nih.gov/pubmed/29436835
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.molpharmaceut.7b01004
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