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Assessing the stability of free-energy perturbation calculations by performing variations in the method

We have calculated relative binding affinities for eight tetrafluorophenyl-triazole-thiogalactoside inhibitors of galectin-3 with the alchemical free-energy perturbation approach. We obtain a mean absolute deviation from experimental estimates of only 2–3 kJ/mol and a correlation coefficient (R(2))...

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Bibliografiske detaljer
Udgivet i:J Comput Aided Mol Des
Main Authors: Manzoni, Francesco, Ryde, Ulf
Format: Artigo
Sprog:Inglês
Udgivet: Springer International Publishing 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5889414/
https://ncbi.nlm.nih.gov/pubmed/29536221
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-018-0110-5
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