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Synthesis of 1,1′-Diarylethanes and Related Systems by Displacement of Trichloroacetimidates with Trimethylaluminum

Benzylic trichloroacetimidates are readily displaced by trimethylaluminum under Lewis acid promoted conditions to provide the corresponding methyl substitution product. This method is a convenient way to access 1,1′-diarylethanes and related systems, which play a significant role in medicinal chemis...

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Detalhes bibliográficos
Publicado no:J Org Chem
Main Authors: Mahajani, Nivedita S., Chisholm, John D.
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5889320/
https://ncbi.nlm.nih.gov/pubmed/29478311
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.8b00027
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