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Biophysical characterization of hit compounds for mechanism-based enzyme activation

Across all families of enzymes, only a dozen or so distinct classes of non-natural small molecule activators have been characterized, with only four known modes of activation among them. All of these modes of activation rely on naturally evolved binding sites that trigger global conformational chang...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:PLoS One
Prif Awduron: Guan, Xiangying, Upadhyay, Alok, Munshi, Sudipto, Chakrabarti, Raj
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: Public Library of Science 2018
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC5856274/
https://ncbi.nlm.nih.gov/pubmed/29547630
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0194175
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