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Numerical analysis of time dependent inhibition kinetics: comparison between rat liver microsomes and rat hepatocyte data for mechanistic model fitting

Time dependent inhibition (TDI) may confound drug interaction predictions. Recently, models were generated for an array of TDI kinetic schemes using numerical analysis of microsomal assays. Additionally, a distinct terminal inactivation step was identified for certain mechanism based inhibitors (MBI...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Xenobiotica
Egile Nagusiak: Pham, Chuong, Nagar, Swati, Korzekwa, Ken
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC5742070/
https://ncbi.nlm.nih.gov/pubmed/28644704
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/00498254.2017.1345020
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