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In vitro binding and receptor-mediated activity of terlipressin at vasopressin receptors V(1) and V(2)

Terlipressin, a synthetic, systemic vasoconstrictor with selective activity at vasopressin-1 (V(1)) receptors, is a pro-drug for the endogenous/natural porcine hormone [Lys(8)]-vasopressin (LVP). We investigated binding and receptor-mediated cellular activities of terlipressin, LVP, and endogenous h...

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Detalles Bibliográficos
Publicado en:J Exp Pharmacol
Main Authors: Jamil, Khurram, Pappas, Stephen Chris, Devarakonda, Krishna R
Formato: Artigo
Idioma:Inglês
Publicado: Dove Medical Press 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5741980/
https://ncbi.nlm.nih.gov/pubmed/29302194
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/JEP.S146034
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