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Synthesis of 1,3-cis-disubstituted sterically encumbered imidazolidinone organocatalysts

A variety of novel imidazolidinone-based organocatalysts with bulky substituents were synthesized under mild reaction conditions starting from easily accessible substrates. Different natural and unnatural amino acid methyl amides were cyclized with aromatic carbaldehydes to yield two diastereomeric...

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Detalhes bibliográficos
Publicado no:Beilstein J Org Chem
Main Authors: Wallbaum, Jan, Werz, Daniel B
Formato: Artigo
Idioma:Inglês
Publicado em: Beilstein-Institut 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5727825/
https://ncbi.nlm.nih.gov/pubmed/29259667
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.13.254
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