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Nonclassical Size Dependence of Permeation Defines Bounds for Passive Adsorption of Large Drug Molecules

Macrocyclic peptides are considered large enough to inhibit “undruggable” targets, but the design of passively cell-permeable molecules in this space remains a challenge due to the poorly understood role of molecular size on passive membrane permeability. Using split-pool combinatorial synthesis, we...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Pye, Cameron R., Hewitt, William M., Schwochert, Joshua, Haddad, Terra D., Townsend, Chad E., Etienne, Lyns, Lao, Yongtong, Limberakis, Chris, Furukawa, Akihiro, Mathiowetz, Alan M., Price, David A., Liras, Spiros, Lokey, R. Scott
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5677520/
https://ncbi.nlm.nih.gov/pubmed/28059508
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b01483
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