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Point mutations affecting antagonist affinity and agonist dependent gating of GABAA receptor channels.

Two variant amino acid sequences, which differ in a single amino acid residue, have been reported for the alpha 1-subunit of the rat brain GABAA receptor. We separately co-expressed these two variants in Xenopus oocytes, in combination with beta 2 and gamma 2. This experiment showed that substitutio...

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Библиографические подробности
Главные авторы: Sigel, E, Baur, R, Kellenberger, S, Malherbe, P
Формат: Artigo
Язык:Inglês
Опубликовано: 1992
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC556666/
https://ncbi.nlm.nih.gov/pubmed/1376242
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