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Characterization of functional μ opioid receptor turnover in rat locus coeruleus: an electrophysiological and immunocytochemical study

BACKGROUND AND PURPOSE: Regulation of μ receptor dynamics such as its trafficking is a possible mechanism underlying opioid tolerance that contributes to inefficient recycling of opioid responses. We aimed to characterize the functional turnover of μ receptors in the noradrenergic nucleus locus coer...

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Publicat a:Br J Pharmacol
Autors principals: Medrano, María Carmen, Santamarta, María Teresa, Pablos, Patricia, Aira, Zigor, Buesa, Itsaso, Azkue, Jon Jatsu, Mendiguren, Aitziber, Pineda, Joseba
Format: Artigo
Idioma:Inglês
Publicat: John Wiley and Sons Inc. 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5522999/
https://ncbi.nlm.nih.gov/pubmed/28589556
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.13901
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