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Population pharmacokinetic and exposure simulation analysis for cediranib (AZD2171) in pooled Phase I/II studies in patients with cancer

AIMS: A population pharmacokinetic (PK) model was developed for cediranib to simulate cediranib exposure for different doses, including comedication with strong uridine glucuronosyl transferase/P‐glycoprotein inducers such as rifampicin, in cancer patients. METHODS: Plasma concentrations and covaria...

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Detalhes bibliográficos
Publicado no:Br J Clin Pharmacol
Main Authors: Li, Jianguo, Al‐Huniti, Nidal, Henningsson, Anja, Tang, Weifeng, Masson, Eric
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5510068/
https://ncbi.nlm.nih.gov/pubmed/28213941
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.13266
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