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A practical and efficient approach to imidazo[1,2-a]pyridine-fused isoquinolines through the post-GBB transformation strategy

Diversity-oriented synthesis of the biologically intriguing imidazo[1,2-a]pyridine-fused isoquinoline systems from readily available starting materials was achieved through the Groebke–Blackburn–Bienaymé reaction followed by a gold-catalyzed cyclization strategy. The synthetic approach is characteri...

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Pubblicato in:Beilstein J Org Chem
Autori principali: Shao, Taofeng, Gong, Zhiming, Su, Tianyi, Hao, Wei, Che, Chao
Natura: Artigo
Lingua:Inglês
Pubblicazione: Beilstein-Institut 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5433183/
https://ncbi.nlm.nih.gov/pubmed/28546839
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.13.82
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