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First total synthesis of concavine

The synthesis of the unusual alkaloid concavine, isolated from Clitocybe concava (Basidiomycetae), has been accomplished. The synthetic route features regio- and stereoselective manipulation of polycyclic imide intermediates via enolate substitution and Grignard addition, along with a key bridge-for...

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Publicat a:Chem Sci
Autors principals: Saint-Dizier, François, Simpkins, Nigel S.
Format: Artigo
Idioma:Inglês
Publicat: Royal Society of Chemistry 2017
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5416908/
https://ncbi.nlm.nih.gov/pubmed/28507709
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6sc05627j
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