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Estimation of relative free energies of binding using pre-computed ensembles based on the single-step free energy perturbation and the site-identification by ligand competitive saturation approaches

Accurate and rapid estimation of relative binding affinities of ligand-protein complexes is a requirement of computational methods for their effective use in rational ligand design. Of the approaches commonly used, free energy perturbation (FEP) methods are considered one of the most accurate, thoug...

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Publicado en:J Comput Chem
Autores principales: Raman, E. Prabhu, Lakkaraju, Sirish Kaushik, Denny, Rajiah Aldrin, MacKerell, Alexander D.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5403604/
https://ncbi.nlm.nih.gov/pubmed/27782307
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jcc.24522
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