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Feasibility and antitumor efficacy in vivo, of simultaneously targeting glycolysis, glutaminolysis and fatty acid synthesis using lonidamine, 6-diazo-5-oxo-L-norleucine and orlistat in colon cancer

The aim of the present study was to investigate in vivo the feasibility and efficacy of the combination of lonidamine (LND), 6-diazo-5-oxo-L-norleucine (DON) and orlistat to simultaneously target glycolysis, glutaminolysis and de novo synthesis of fatty acids, respectively. The doses of LND and DON...

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Dettagli Bibliografici
Pubblicato in:Oncol Lett
Autori principali: Cervantes-Madrid, Diana, Dominguez-Gomez, Guadalupe, Gonzalez-Fierro, Aurora, Perez-Cardenas, Enrique, Taja-Chayeb, Lucia, Trejo-Becerril, Catalina, Duenas-Gonzalez, Alfonso
Natura: Artigo
Lingua:Inglês
Pubblicazione: D.A. Spandidos 2017
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5403504/
https://ncbi.nlm.nih.gov/pubmed/28454342
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3892/ol.2017.5615
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