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The Development of CK2 Inhibitors: From Traditional Pharmacology to in Silico Rational Drug Design

Casein kinase II (CK2) is an ubiquitous and pleiotropic serine/threonine protein kinase able to phosphorylate hundreds of substrates. Being implicated in several human diseases, from neurodegeneration to cancer, the biological roles of CK2 have been intensively studied. Upregulation of CK2 has been...

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Detaylı Bibliyografya
Yayımlandı:Pharmaceuticals (Basel)
Yazar: Cozza, Giorgio
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: MDPI 2017
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC5374430/
https://ncbi.nlm.nih.gov/pubmed/28230762
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph10010026
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