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Combatting AMR: photoactivatable ruthenium(ii)-isoniazid complex exhibits rapid selective antimycobacterial activity

The novel photoactive ruthenium(ii) complex cis-[Ru(bpy)(2)(INH)(2)][PF(6)](2) (1·2PF(6), INH = isoniazid) was designed to incorporate the anti-tuberculosis drug, isoniazid, that could be released from the Ru(ii) cage by photoactivation with visible light. In aqueous solution, 1 rapidly released two...

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Argitaratua izan da:Chem Sci
Egile Nagusiak: Smith, Nichola A., Zhang, Pingyu, Greenough, Simon E., Horbury, Michael D., Clarkson, Guy J., McFeely, Daniel, Habtemariam, Abraha, Salassa, Luca, Stavros, Vasilios G., Dowson, Christopher G., Sadler, Peter J.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Royal Society of Chemistry 2017
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Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC5365061/
https://ncbi.nlm.nih.gov/pubmed/28451184
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6sc03028a
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