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Zirconium tetraazamacrocycle complexes display extraordinary stability and provide a new strategy for zirconium-89-based radiopharmaceutical development

We report our initial investigations into the use of tetraazamacrocycles as zirconium-89 chelators. We describe the synthesis and complete characterization of several Zr tetraazamacrocycle complexes, and definitively describe the first crystal structure of zirconium 1,4,7,10-tetraazacyclododecane-1,...

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Detalhes bibliográficos
Publicado no:Chem Sci
Main Authors: Pandya, Darpan N., Bhatt, Nikunj, Yuan, Hong, Day, Cynthia S., Ehrmann, Brandie M., Wright, Marcus, Bierbach, Ulrich, Wadas, Thaddeus J.
Formato: Artigo
Idioma:Inglês
Publicado em: Royal Society of Chemistry 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5363373/
https://ncbi.nlm.nih.gov/pubmed/28451334
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6sc04128k
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