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Functional, electrophysiological and molecular docking analysis of the modulation of Ca(v)1.2 channels in rat vascular myocytes by murrayafoline A

BACKGROUND AND PURPOSE: The carbazole alkaloid murrayafoline A (MuA) enhances contractility and the Ca(2+) currents carried by the Ca(v)1.2 channels [I(Ca1.2)] of rat cardiomyocytes. As only few drugs stimulate I(Ca1.2), this study was designed to analyse the effects of MuA on vascular Ca(v)1.2 chan...

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Библиографические подробности
Опубликовано в: :Br J Pharmacol
Главные авторы: Saponara, S, Durante, M, Spiga, O, Mugnai, P, Sgaragli, G, Huong, TT, Khanh, PN, Son, NT, Cuong, NM, Fusi, F
Формат: Artigo
Язык:Inglês
Опубликовано: John Wiley and Sons Inc. 2016
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5341225/
https://ncbi.nlm.nih.gov/pubmed/26493241
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.13369
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