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In silico analysis of the binding of anthelmintics to Caenorhabditis elegansP-glycoprotein 1

Macrocyclic lactones (ML) are important anthelmintics used in animals and humans against parasite nematodes, but their therapeutic success is compromised by the spread of ML resistance. Some ABC transporters, such as p-glycoproteins (Pgps), are selected and overexpressed in ML-resistant nematodes, s...

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Detalhes bibliográficos
Publicado no:Int J Parasitol Drugs Drug Resist
Main Authors: David, Marion A., Orlowski, Stéphane, Prichard, Roger K., Hashem, Shaima, André, François, Lespine, Anne
Formato: Artigo
Idioma:Inglês
Publicado em: Elsevier 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5196494/
https://ncbi.nlm.nih.gov/pubmed/27746191
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijpddr.2016.09.001
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